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New Synthetic Isoxazole Derivatives Acting as Potent Inducers of Fetal Hemoglobin in Erythroid Precursor Cells Isolated from β-Thalassemic Patients Zuccato, Cristina; Cosenza, Lucia Carmela; Tupini, Chiara; Finotti, Alessia; Sacchetti, Gianni; Simoni, Daniele; Gambari, Roberto; Lampronti, Ilaria dettagli >>	MOLECULES Vol. 29, No. 1, pp: 8-1-8-16, Anno: 2024

Pro‑apoptotic activity of novel synthetic isoxazole derivatives exhibiting inhibitory activity against tumor cell growth in vitro Lampronti, I.; Simoni, D.; Rondanin, R.; Baruchello, R.; Scapoli, C.; Finotti, A.; Borgatti, M.; Tupini, C.; Gambari, R. dettagli >>	ONCOLOGY LETTERS Vol. 20, No. 5, pp: 151-1-151-11, Anno: 2020

New TRAP1 and Hsp90 chaperone inhibitors with cationic components: Preliminary studies on mitochondrial targeting Rondanin, R; Lettini, G; Oliva, P; Baruchello, R; Costantini, C; Trapella, C; Simoni, D; Bernardi, T; Sisinni, L; Pietrafesa, M; Ponterini, G; Costi, M P; Vignudelli, T; Luciani, R; Matassa, D S; Esposito, F; Landriscina, M dettagli >>	BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS Vol. 28, No. 13, pp: 2289-2293, Anno: 2018

Effects of Pimozide Derivatives on pSTAT5 in K562 Cells Rondanin, Riccardo; Simoni, Daniele; Maccesi, Martina; Romagnoli, Romeo; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Cascio, Antonio; Tolomeo, Manlio dettagli >>	CHEMMEDCHEM Vol. 12, No. 15, pp: 1183-1190, Anno: 2017

Arylamidonaphtalene sulfonate compounds as a novel class of heparanase inhibitors Rondanin, Riccardo; Fochi, Sara; Baruchello, Riccardo; Bernardi, Tatiana; Oliva, Paola; Semeraro, Floriana; Simoni, Daniele; Giannini, Giuseppe dettagli >>	BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS Vol. 27, No. 18, pp: 4421-4425, Anno: 2017

Novel iodoacetamido benzoheterocyclic derivatives with potent antileukemic activity are inhibitors of STAT5 phosphorylation Romagnoli, Romeo; Baraldi, Pier Giovanni; Prencipe, Filippo; Lopez Cara, Carlota; Rondanin, Riccardo; Simoni, Daniele; Hamel, Ernest; Grimaudo, Stefania; Pipitone, Rosaria Maria; Meli, Maria; Tolomeo, Manlio dettagli >>	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY Vol. 108, No. 1, pp: 39-52, Anno: 2016

Hemiasterlin derivative (R)(S)(S)-BF65 and Akt inhibitor MK-2206 synergistically inhibit SKOV3 ovarian cancer cell growth Lai, Wei Ting; Cheng, Kai Lin; Baruchello, Riccardo; Rondanin, Riccardo; Marchetti, Paolo; Simoni, Daniele; Lee, Ray M.; Guh, Jih Hwa; Hsu, Lih Ching dettagli >>	BIOCHEMICAL PHARMACOLOGY Vol. 113, No. 1, pp: 12-23, Anno: 2016

A novel hybrid drug between two potent anti-tubulin agents as a potential prolonged anticancer approach Marchetti, Paolo; Pavan, Barbara; Simoni, Daniele; Baruchello, Riccardo; Rondanin, Riccardo; Mischiati, Carlo; Feriotto, Giordana; Ferraro, Luca Nicola; Hsu, Lih Ching; Lee, Ray M.; Dalpiaz, Alessandro dettagli >>	EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES Vol. 91, No. 1, pp: 50-63, Anno: 2016

Inhibition of activated STAT5 in Bcr/Abl expressing leukemia cells with new pimozide derivatives. Rondanin, Riccardo; Simoni, Daniele; Romagnoli, Romeo; Baruchello, Riccardo; Marchetti, Paolo; Costantini, Cristiana; Fochi, Sara; Padroni, Giacomo; S., Grimaudo; R. M., Pipitone; M., Meli; M., Tolomeo dettagli >>	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 24, No. 1, pp: 4568-4574, Anno: 2014

4,5,6,7-Tetrahydro-isoxazolo-[4,5-c]-pyridines as a new class of cytotoxic Hsp90 inhibitors Baruchello, Riccardo; Simoni, Daniele; Marchetti, Paolo; Rondanin, Riccardo; Mangiola, Stefania; Costantini, Cristiana; M., Meli; G., Giannini; L., Vesci; V., Carollo; T., Brunetti; G., Battistuzzi; M., Tolomeo; W., Cabri dettagli >>	EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY Vol. 76, No. 1, pp: 53-60, Anno: 2014

Stilbene 5c, a microtubule poison with vascular disrupting properties that induces multiple modes of growth arrest and cell death. M. R., Alotaibi; B., Asnake; X., Di; M. J., Beckman; D., Durrant; Simoni, Daniele; Baruchello, Riccardo; R. M., Lee; E. L., Schwartz; D. A., Gewirtz dettagli >>	BIOCHEMICAL PHARMACOLOGY Vol. 86, No. 1, pp: 1688-1698, Anno: 2013

The new iodoacetamidobenzofuran derivative TR120 decreases STAT5 expression and induces antitumor effects in imatinib-sensitive and imatinib-resistant BCR-ABL-expressing leukemia cells Grimaudo, S.; Meli, M.; Di Cristina, A.; Ferro, A.; Pipiton, M. R.; Romagnoli, Romeo; Simoni, Daniele; Dieli, F.; Tolomeo, M. dettagli >>	ANTI-CANCER DRUGS Vol. 24, No. 4, pp: 384-393, Anno: 2013

Development of hemiasterlin derivatives as potential anticancer agents that inhibit tubulin polymerization and synergize with a stilbene tubulin inhibitor. L., Hsu; D. E., Durrant; C., Huang; N., Chi; Baruchello, Riccardo; Rondanin, Riccardo; Rullo, Cinzia; Marchetti, Paolo; Grisolia, Giuseppina; Simoni, Daniele; R. M., Lee dettagli >>	INVESTIGATIONAL NEW DRUGS Vol. 30, No. 1, pp: 1379-1388, Anno: 2012

Synthesis and biological activity of a novel class nicotinic acetylcholine receptors (nAChRs) ligands structurally related to anatoxin-a. Simoni, Daniele; Rondanin, Riccardo; Marchetti, Paolo; Rullo, Cinzia; Baruchello, Riccardo; Grisolia, Giuseppina; G., Barbato; R., Giovannini; C., Marchioro; A. M., Capelli; C., Virginio; A., Bozzoli; Borea, Pier Andrea; Merighi, Stefania; D., Donati dettagli >>	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 21, No. 1, pp: 5423-5427, Anno: 2011

Novel 3,4-isoxazolediamides as potent inhibitors of chaperone heat shock protein 90. Baruchello, Riccardo; Simoni, Daniele; Grisolia, Giuseppina; G., Barbato; Marchetti, Paolo; Rondanin, Riccardo; Mangiola, Stefania; G., Giannini; T., Brunetti; D., Alloatti; G., Gallo; A., Ciacci; L., Vesci; M., Castorina; F. M., Milazzo; M. L., Cervoni; M. B., Guglielmi; M., Barbarino; R., Foderà; C., Pisano; W., Cabri dettagli >>	JOURNAL OF MEDICINAL CHEMISTRY Vol. 54, No. 1, pp: 8592-8604, Anno: 2011

Versatile Synthesis of New Cytotoxic Agents Structurally Related to Emiasterlins Simoni, Daniele; R. M., Lee; D. E., Durrant; N., Chi; Baruchello, Riccardo; Rondanin, Riccardo; Rullo, Cinzia; Marchetti, Paolo dettagli >>	BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Vol. 20, No. 1, pp: 3431-3435, Anno: 2010

Tyrosine kinase ihibitors for the treatment of chronic myeloid leukemia M., Tolomeo; F., Dieli; N., Gebbia; Simoni, Daniele dettagli >>	ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY Vol. 9, No. 8, pp: 853-863, Anno: 2009

Hydropathic analysis and biological evaluation of stilbene derivatives as colchicine site microtubule inhibitors with anti-leukemic activity. A., Tripathi; D., Durrant; R. M., Lee; Baruchello, Riccardo; Romagnoli, Romeo; Simoni, Daniele; G. E., Kellogg dettagli >>	JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Vol. 24, No. 6, pp: 1237-1244, Anno: 2009

Development of water soluble derivatives of cis-3, 4', 5-trimethoxy-3'-aminostilbene for optimization and use in cancer therapy. David E., Durrant; Joanna, Richards; Ashutosh, Tripathi; Glen E., Kellogg; Marchetti, Paolo; Eleopra, Marco; Grisolia, Giuseppina; Simoni, Daniele; Ray M., Lee dettagli >>	INVESTIGATIONAL NEW DRUGS Vol. 27, No. 1, pp: 41-52, Anno: 2009

Design, synthesis and biological evaluation of novel stilbene-based antitumor agents Simoni, Daniele; Francesco Paolo, Invidiata; Eleopra, Marco; Marchetti, Paolo; Rondanin, Riccardo; Baruchello, Riccardo; Grisolia, Giuseppina; Ashutosh, Tripathi; Glen E., Kellogg; David, Durrant; Ray M., Lee dettagli >>	BIOORGANIC & MEDICINAL CHEMISTRY Vol. 17, No. 2, pp: 512-522, Anno: 2009